Non-Effective Improvement of Absorption for Some Nanoparticle Formulations Explained by Permeability under Non-Sink Conditions

We evaluated the in vitro permeability of nanoparticle formulations of high and low lipophilic compounds under non-sink conditions, wherein compounds are not completely dissolved. The permeability of the highly lipophilic compound, griseofulvin, was improved by about 30% due to nanonization under no...

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Главные авторы: Kazuya Sugita (Автор), Noriyuki Takata (Автор), Etsuo Yonemochi (Автор)
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Опубликовано: MDPI AG, 2022-04-01T00:00:00Z.
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