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Enantioselective Synthesis and Pharmacological Evaluation of Aza-CGP37157-Lipoic Acid Hybrids for the Treatment of Alzheimer's Disease

Hybrids based on an aza-analogue of CGP37157, a mitochondrial Na<sup>+</sup>/Ca<sup>2+</sup> exchanger antagonist, and lipoic acid were obtained in order to combine in a single molecule the antioxidant and NRF2 induction properties of lipoic acid and the neuroprotective activ...

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Main Authors:	Ángel Cores (Author), Patrycja Michalska (Author), José Miguel Pérez (Author), Enrique Crisman (Author), Clara Gómez (Author), Mercedes Villacampa (Author), José Carlos Menéndez (Author), Rafael León (Author)
Format:	Book
Published:	MDPI AG, 2022-01-01T00:00:00Z.
Subjects:	article
Online Access:	Connect to this object online.
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