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Screening of benzenesulfonamide in combination with chemically diverse fragments against carbonic anhydrase by differential scanning fluorimetry

The differential scanning fluorimetry (DSF) screening of 5.692 fragments in combination with benzenesulfonamide (BSA) against bovine carbonic anhydrase (bCA) delivered >100 hits that either caused, on their own, a significant thermal shift (ΔTm, °C) in the protein melting temperature or significa...

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Main Authors:	Mikhail Krasavin (Author), Stanislav Kalinin (Author), Sergey Zozulya (Author), Anastasiia Gryniukova (Author), Petro Borysko (Author), Andrea Angeli (Author), Claudiu T. Supuran (Author)
Format:	Book
Published:	Taylor & Francis Group, 2020-01-01T00:00:00Z.
Subjects:	article
Online Access:	Connect to this object online.
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